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Remoxipride hydrochloride
CAS No. 73220-03-8
Remoxipride hydrochloride( Roxiam | (S)-Remoxipride Hydrochloride | Remoxipride Hydrochloride Anhydrous )
Catalog No. M27695 CAS No. 73220-03-8
Dopamine D2 receptor antagonist.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 107 | Get Quote |
|
| 5MG | 160 | Get Quote |
|
| 10MG | 194 | Get Quote |
|
| 25MG | 428 | Get Quote |
|
| 50MG | 626 | Get Quote |
|
| 100MG | 889 | Get Quote |
|
| 500MG | 1782 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameRemoxipride hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionDopamine D2 receptor antagonist.
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DescriptionDopamine D2 receptor antagonist.(In Vivo):In male Sprague-Dawley rats, Remoxipride hydrochloride (0.1-100 μM/kg; i.p.) blockes apomorphine-induced hyperactivity and dose-dependent blockades apomorphine-induced behaviors. In beagle dogs, Remoxipride hydrochloride (0.25-5 μM/kg; gavage) blockes apomorphine-induced vomiting.
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In Vitro(S)-Remoxipride hydrochloride (1-100 μM; 20 min) shows binding efficiency with IC50s of ＞100, 1.57 and 42 μM for dopamine D1, dopamine D2 and α1-Adrenoccptor, respectively.
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In Vivo(S)-Remoxipride hydrochloride (0.1-100 μM/kg; i.p. 60 min prior to apomorphine) blockades apomorphine-induced behaviors s in rats and vomiting in dogs.(S)-Remoxipride hydrochloride (0.1-10 mg/kg; i.p. 30 min prior to apomorphine) displaces [3H]spiperone from both striatal and extra-striatal areas.
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SynonymsRoxiam | (S)-Remoxipride Hydrochloride | Remoxipride Hydrochloride Anhydrous
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PathwayOthers
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TargetOther Targets
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number73220-03-8
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Formula Weight407.73
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Molecular FormulaC16H24BrClN2O3
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Purity>98% (HPLC)
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Solubility——
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SMILESCl.CCN1CCC[C@H]1CNC(=O)c1c(OC)ccc(Br)c1OC
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Richard W. Watkins, et al. Evaluation of cinnamamide as an avian repellent: Determination of a dose—response curve.
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